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Bretazenil用途是什么?

提问时间:2021/9/9 14:29:44

描述:Bretazenil是做什么用的?哪里可以用到Bretazenil?

admin 2021-09-09 14:29
Bretazenil溴他西尼用途Bretazenil, also known as Ro 16-6028, is GABA A receptor agonist potentially for the treatment of anxiety disorders. Bretazenil differs from traditional 1,4-benzodiazepines by being a partial agonist and because it binds to α1, α2, α3, α4, α5 and α6 subunit containing GABAA receptor benzodiazepine receptor complexes. 1,4-benzodiazepines bind only to α1, α2, α3 and α5 GABAA benzodiazepine receptor complexes.

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